GW501516 (Cardarine) – 20mg/ml Liquid

GW501516 is a selective agonist of the PPARδ receptor that displays high affinity and potency for PPARδ with > 1,000 fold selectivity over PPARα and PPARγ. In rats, binding of GW501516 to PPARδ recruits the coactivator PGC-1α . It was initially discovered during a research collaboration between GSK and Ligand Pharmaceuticals that began in 1992  The drug entered into clinical development as a drug candidate for metabolic and cardiovascular diseases, but was abandoned in 2007 because animal testing showed that the drug caused cancer to develop rapidly in several organs

Specifications

• Chemical Formula: C21H18F3NO3S2
• Molecular Mass: 453.50 g/mol
• Synonyms: GSK 516, GW1516, GW 501516, GW 501,516, Cardarine
• CAS Number: 317318-70-0
• PubChem: 9803963
• Total Amount of the Active Ingredient: 20 mg/ml
• Shelf Life: 36 months